PSMA617，1702967-37-0，一种化学修饰的 PSMA抑制剂

文章关键词：1702967-37-0，PSMA617， Vipivotide tetraxetan

一、基本信息

【性质简介】：PSMA-617 has enhanced its targeting ability towards PSMA through a series of precise chemical modifications. The Ki value, as an important indicator of the binding ability between drugs and targets, is only 0.37 nM for PSMA-617. The breakthrough in this value means that the binding ability between drugs and PSMA has reached an unprecedented height. The emergence of PSMA-617 undoubtedly brings new hope to cancer patients with high expression of PSMA, such as prostate cancer. Its high specificity enables drugs to kill tumor cells more accurately while maximizing the protection of normal cells from damage. In addition, the excellent pharmacokinetic properties of PSMA-617 have laid a solid foundation for its widespread promotion in clinical applications. PSMA-617 has shown great potential in the field of cancer treatment due to its excellent PSMA inhibition ability and low Ki value.

【英文名】：PSMA617， Vipivotide tetraxetan

【CAS号】：1702967-37-0

【化学式】：C49H71N9O16

【分子量】：1042.14

【结构式】：

 

​二、详情介绍

【外观】：固体/粉末

【溶解性】：溶于大部分有机溶剂

【规格】：1g、5g、10g

【纯度】：95%+

【储存条件】：本品应密封避光，储存于阴凉、干燥、通风处，避免反复冻融，储液应该立即使用

【注意事项】：试剂仅用于科学研究或者工业应用等非医疗目的，非药用，非食用！

三、相关试剂

（Sulfo-Cyanine3-DA）磺化-Cy3-多巴胺

（Sulfo-Cyanine3-Resveratrol）磺化-Cy3-白藜芦醇

（Sulfo-Cy3-IHR）磺化-Cy3-IHR

（Sulfo-Cy3-dCTP）磺化-Cy3-dCTP

（Sulfo-Cy3-Methyltetrazine） 磺化-Cy3-甲氧基四嗪

（Sulfo-Cyanine3-hydrazide）磺化-Cy3-酰肼

（Sulfo-Cy3-aldehyde） 磺化-Cy3-醛

（Cyanine3-DA）Cy3-多巴胺

（Sulfo-Cy3-HAIYPRH）Sulfo-Cy3-转铁蛋白靶向肽

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