环肽抑制剂：1088715-84-7，LY2510924，LY2510924游离态，试剂相关特点说明

​编辑资料作者：陕西新研博美生物科技有限公司小编MISSwu​

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LY2510924，LY2510924游离态，拮抗剂LY2510924，环肽，抑制剂

Product structure：

Product specifications：
1.CAS No：1088715-84-7
2.Molecular formula：C62H88N14O10
3.Molecular weight：1189.450
4.density：1.3±0.1 g/cm3
5.Packaging specification：1g、5g、10g, flexible packaging, including 100mg packaging and 500mg 1g and 5g large packaging
6.Dissolution conditions：Soluble in most organic solvents, such as DCM, DMF, DMSO, THF, etc., with good solubility in water
7.Stability：-1 year at 20 ° C, dry and dark.
Reaction characteristics：
LY2510924是一种有效的、选择性的CXCR4拮抗剂，特异性地阻止SDF-1与CXCR4的结合，IC50为0.079 nM；抑制SDF-1诱导的GTP结合，Kb值为0.38 nM。

LY2510924抑制SDF-1诱导的细胞迁移，IC50为0.26 nM；并抑制SDF-1/CXCR4介导的胞内信号。LY2510924没有明显的激动活性。它对其他趋化因子受体如CCR1,CCR2,CXCR2和CXCRChemicalbook3在检测浓度下没有抑制活性，对5-羟色胺受体、多巴胺受体、opioidreceptors也没有活性。

Matters for use：
It is sensitive to light and temperature. In order to use the reagent effectively, the material should always be kept in a low temperature dry condition, away from light, and avoid frequent thawing and freezing.
storage conditions:
Store at - 20 ℃ as much as possible. If conditions permit, the material can be treated under inert gas to obtain better stability of the reagent.
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以上编辑的试剂信息仅用于科学研究或者工业应用等非医疗目的，非药用，非食用。接受各种复杂定制服务，合成的Monodispersed PEGs除了有更多样的基团还可以提供各种不同数量的PEG的产品。