MCE 国际站:naUbrogepantc
参考详情:Ubrogepant (MK-1602,乌布吉泮) - 仅供科研 | CGRP拮抗剂 | MCE
CAS:1374248-77-7
品牌:MedChemExpress (MCE)
存储条件:Powder: -20°C, 3 years; 4°C, 2 years.In solvent: -80°C, 6 months; -20°C, 1 month.
生物活性:Ubrogepant (MK-1602) 是一种新型口服降钙素基因相关肽受体 (CGRP) 拮抗剂,正在开发用于急性偏头痛的治疗[1]。 IC50 和目标:MK-1602[1]
热销产品:Olutasidenib | GR24 | 1,2-Distearoyl-sn-glycero-3-phosphorylcholine-d70 | HUHS015 | PEG6000 | Stearamide | Alpha-2-macroglobulin, Human (sf9, His) | Flavokawain A | Topiramate | Simethicone
研究领域:GPCR/G Protein | Neuronal Signaling
作用靶点:CGRP Receptor
Trending products:Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Fluorescent Dye | PROTAC | Isotope-Labeled Compounds | Oligonucleotides
参考文献:
[1]. Li CC, et al. Population PK Analyses of Ubrogepant (MK-1602), a CGRP Receptor Antagonist: Enriching In-Clinic Plasma PK Sampling With Outpatient Dried Blood Spot Sampling. J Clin Pharmacol. 2017 Nov 14. doi: 10.1002/jcph.1021.